12 patents
Utility
BRM targeting compounds and associated methods of use
18 Jul 23
The present disclosure provides bifunctional compounds comprising a target protein binding moiety and a E3 ubiquitin ligase binding moiety, and associated methods of use.
Hong Lin, Philip Pitis, Liang Lu, Andrew Paul Combs
Filed: 9 Jun 21
Utility
CDK inhibitors and their use as pharmaceuticals
27 Jun 23
Andrew W. Buesking, Andrew Paul Combs, Jincong Zhuo, Ryan Holmes, Sarah Pawley, Xiaowei Wu
Filed: 21 Sep 21
Utility
BCL-2 inhibitors and their use as pharmaceuticals
11 Apr 23
The disclosure is directed to, in part, to BCL-2 inhibitors, pharmaceutical compositions comprising the same, as well as methods of their use and preparation.
Jincong Zhuo, Andrew Paul Combs, Peng Wei, Jialiang Wang
Filed: 27 Apr 21
Utility
Substituted pyrrolo[2,3-d]pyrimidines as inhibitors of protein arginine methyl transferase 5 (PRMT5)
13 Dec 22
Juan Luengo, Hong Lin, Michael Hawkins
Filed: 26 Oct 18
Utility
Selective inhibitors of protein arginine methyltransferase 5 (PRMT5)
22 Feb 22
Juan Luengo, Hong Lin, Michael Hawkins, Rupa Shetty, Philip Pitis, Gisela Saborit Villarroya
Filed: 5 Aug 20
Utility
Selective inhibitors of protein arginine methyltransferase 5 (PRMT5)
11 Jan 22
Juan Luengo, Raul A. Leal, Hong Lin, Rupa Shetty, Krishna Vaddi
Filed: 20 Feb 18
Utility
Selective inhibitors of protein arginine methyltransferase 5 (PRMT5)
4 Jan 22
Juan Luengo, Hong Lin, Michael Hawkins, Rupa Shetty, Philip Pitis, Gisela Saborit Villarroya
Filed: 1 Jun 20
Utility
Selective inhibitors of protein arginine methytransterase 5 (PRMT5)
28 Dec 21
Hong Lin, Juan Luengo, Rupa Shetty, Michael Hawkins
Filed: 5 Aug 20
Utility
Spiro-sulfonamide derivatives as inhibitors of myeloid cell leukemia-1 (MCL-1) protein
28 Sep 21
Jincong Zhuo, Raul Leal, Rupa Shetty, Juan Luengo, Andrew Paul Combs, Peng Wei
Filed: 8 Nov 19
Utility
Selective inhibitors of protein arginine methlytransferase 5 (PRMT5)
3 Aug 21
Hong Lin, Juan Luengo, Rupa Shetty, Michael Hawkins
Filed: 16 Jan 20
Utility
Selective inhibitors of protein arginine methyltransferase 5 (PRMT5)
13 Jul 20
Juan Luengo, Hong Lin, Michael Hawkins, Rupa Shetty, Philip Pitis, Gisela Saborit Villarroya
Filed: 4 Apr 19
Utility
Selective inhibitors of protein arginine methyltransferase 5 (PRMT5)
24 Feb 20
Hong Lin, Juan Luengo, Rupa Shetty, Michael Hawkins
Filed: 8 Aug 18
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